Discovery of a phenylpyrazole amide ROCK inhibitor as a tool molecule for in vivo studies

Hu Z, Wang C, Glunz PW, Li J, Cheadle NL, Chen AY, Chen X-Q, Myers JE, Guarino VR, Rose A, Sack JS, Sitkoff D, Taylor DS, Xu S, Yan C, Zhang H, Zhang L, Hennan J, Adam LP, Wexler RR & Quan ML
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Hu, Z., Wang, C., Glunz, P. W., Li, J., Cheadle, N. L., Chen, A. Y., … Quan, M. L. (2020). Discovery of a phenylpyrazole amide ROCK inhibitor as a tool molecule for in vivo studies. Bioorganic and Medicinal Chemistry Letters, 30(21), 127495 (4 pp.). https://doi.org/10.1016/j.bmcl.2020.127495