Structure-based and property-driven optimization of N-aryl imidazoles toward potent and selective oral RORγt inhibitors

Hoegenauer K, Kallen J, Jiménez-Núñez E, Strang R, Ertl P, Cooke NG, Hintermann S, Voegtle M, Betschart C, McKay DJJ, Wagner J, Ottl J, Beerli C, Billich A, Dawson J, Kaupmann K, Streiff M, Gobeau N, Harlfinger S, Stringer R & Guntermann C
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Hoegenauer, K., Kallen, J., Jiménez-Núñez, E., Strang, R., Ertl, P., Cooke, N. G., … Guntermann, C. (2019). Structure-based and property-driven optimization of N-aryl imidazoles toward potent and selective oral RORγt inhibitors. Journal of Medicinal Chemistry, 62(23), 10816-10832. https://doi.org/10.1021/acs.jmedchem.9b01291