Discovery of potent, highly selective, and in vivo efficacious, allosteric MALT1 inhibitors by iterative scaffold morphing

Pissot Soldermann C, Simic O, Renatus M, Erbel P, Melkko S, Wartmann M, Bigaud M, Weiss A, McSheehy P, Endres R, Santos P, Blank J, Schuffenhauer A, Bold G, Buschmann N, Zoller T, Altmann E, Manley PW, Dix I, Buchdunger E, Scesa J, Quancard J, Schlapbach A, Bornancin F, Radimerski T & Régnier CH
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Pissot Soldermann, C., Simic, O., Renatus, M., Erbel, P., Melkko, S., Wartmann, M., … Régnier, C. H. (2020). Discovery of potent, highly selective, and in vivo efficacious, allosteric MALT1 inhibitors by iterative scaffold morphing. Journal of Medicinal Chemistry, 63(23), 14576-14593. https://doi.org/10.1021/acs.jmedchem.0c01245