Active Filters

  • (-) Publication Year = 2021
  • (-) Publication Types = Journal Article
  • (-) Full Text: Restricted OR Full Text: No Full Text
  • (-) Collection = *:external
  • (-) Journals = Bioorganic and Medicinal Chemistry Letters
Search Results 1 - 4 of 4
  • RSS Feed
Select Page
Discovery of a new series of PI3K-δ inhibitors from virtual screening
Fradera, X., Deng, Q., Achab, A., Garcia, Y., Kattar, S. D., McGowan, M. A., … Katz, J. D. (2021). Discovery of a new series of PI3K-δ inhibitors from virtual screening. Bioorganic and Medicinal Chemistry Letters, 42, 128046 (5 pp.). https://doi.org/10.1016/j.bmcl.2021.128046
Discovery and optimization of covalent EGFR T790M/L858R mutant inhibitors
Hoogenboom, N., Demont, D., de Zwart, E., Verkaik, S., Emmelot, M., van de Kar, B., … Barf, T. (2021). Discovery and optimization of covalent EGFR T790M/L858R mutant inhibitors. Bioorganic and Medicinal Chemistry Letters, 52, 128406 (6 pp.). https://doi.org/10.1016/j.bmcl.2021.128406
Development of autotaxin inhibitors: a series of tetrazole cinnamides
Thomson, C. G., Le Grand, D., Dowling, M., Beattie, D., Elphick, L., Faller, M., … Zink, F. (2021). Development of autotaxin inhibitors: a series of tetrazole cinnamides. Bioorganic and Medicinal Chemistry Letters, 31, 127663 (7 pp.). https://doi.org/10.1016/j.bmcl.2020.127663
Novel bicyclic pyrazoles as potent ALK2 (R206H) inhibitors for the treatment of fibrodysplasia ossificans progressiva
Yamamoto, H., Sakai, N., Ohte, S., Sato, T., Sekimata, K., Matsumoto, T., … Koyama, H. (2021). Novel bicyclic pyrazoles as potent ALK2 (R206H) inhibitors for the treatment of fibrodysplasia ossificans progressiva. Bioorganic and Medicinal Chemistry Letters, 38, 127858 (5 pp.). https://doi.org/10.1016/j.bmcl.2021.127858