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Discovery of LOU064 (remibrutinib), a potent and highly selective covalent inhibitor of Bruton's tyrosine kinase
Angst, D., Gessier, F., Janser, P., Vulpetti, A., Wälchli, R., Beerli, C., … Cenni, B. (2020). Discovery of LOU064 (remibrutinib), a potent and highly selective covalent inhibitor of Bruton's tyrosine kinase. Journal of Medicinal Chemistry. https://doi.org/10.1021/acs.jmedchem.9b01916
The ABC exporter IrtAB imports and reduces mycobacterial siderophores
Arnold, F. M., Weber, M. S., Gonda, I., Gallenito, M. J., Adenau, S., Egloff, P., … Seeger, M. A. (2020). The ABC exporter IrtAB imports and reduces mycobacterial siderophores. Nature, 580(7803), 413-417. https://doi.org/10.1038/s41586-020-2136-9
Structures in tetrahydrofolate methylation in desulfitobacterial glycine betaine metabolism at atomic resolution
Badmann, T., & Groll, M. (2020). Structures in tetrahydrofolate methylation in desulfitobacterial glycine betaine metabolism at atomic resolution. ChemBioChem, 21(6), 776-779. https://doi.org/10.1002/cbic.201900515
On-surface synthesis of nonmetal porphyrins
Baklanov, A., Garnica, M., Robert, A., Bocquet, M. L., Seufert, K., Küchle, J. T., … Auwärter, W. (2020). On-surface synthesis of nonmetal porphyrins. Journal of the American Chemical Society, 142(4), 1871-1881. https://doi.org/10.1021/jacs.9b10711
Mechanisms of regulation and diverse activities of tau-tubulin kinase (TTBK) isoforms
Bao, C., Bajrami, B., Marcotte, D. J., Chodaparambil, J. V., Kerns, H. M., Henderson, J., … Dillon, G. M. (2020). Mechanisms of regulation and diverse activities of tau-tubulin kinase (TTBK) isoforms. Cellular and Molecular Neurobiology. https://doi.org/10.1007/s10571-020-00875-6
Targeting cavity-creating p53 cancer mutations with small-molecule stabilizers: the Y220X paradigm
Bauer, M. R., Krämer, A., Settanni, G., Jones, R. N., Ni, X., Khan Tareque, R., … Joerger, A. C. (2020). Targeting cavity-creating p53 cancer mutations with small-molecule stabilizers: the Y220X paradigm. ACS Chemical Biology, 15(3), 657-668. https://doi.org/10.1021/acschembio.9b00748
Structural basis for the recognition of transiently structured AU-rich elements by Roquin
Binas, O., Tants, J. N., Peter, S. A., Janowski, R., Davydova, E., Braun, J., … Schlundt, A. (2020). Structural basis for the recognition of transiently structured AU-rich elements by Roquin. Nucleic Acids Research. https://doi.org/10.1093/nar/gkaa465
Identification of FAM181A and FAM181B as new interactors with the TEAD transcription factors
Bokhovchuk, F., Mesrouze, Y., Delaunay, C., Martin, T., Villard, F., Meyerhofer, M., … Chène, P. (2020). Identification of FAM181A and FAM181B as new interactors with the TEAD transcription factors. Protein Science, 29(2), 509-520. https://doi.org/10.1002/pro.3775
'Drc', a structurally novel ssDNA-binding transcription regulator of N4-related bacterial viruses
Boon, M., De Zitter, E., De Smet, J., Wagemans, J., Voet, M., Pennemann, F. L., … Lavigne, R. (2020). 'Drc', a structurally novel ssDNA-binding transcription regulator of N4-related bacterial viruses. Nucleic Acids Research, 48(1), 445-459. https://doi.org/10.1093/nar/gkz1048
Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity
Borreschmidt Hansen, B., Jepsen, T. H., Larsen, M., Sindet, R., Vifian, T., Nørreskov Burhardt, M., … Ritzén, A. (2020). Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity. Journal of Medicinal Chemistry. https://doi.org/10.1021/acs.jmedchem.0c00359
Modulation of the <em>Erwinia </em>ligand-gated ion channel (ELIC) and the 5-HT<sub>3</sub> receptor via a common vestibule site
Brams, M., Govaerts, C., Kambara, K., Price, K. L., Spurny, R., Gharpure, A., … Ulens, C. (2020). Modulation of the Erwinia ligand-gated ion channel (ELIC) and the 5-HT3 receptor via a common vestibule site. eLife, 9, e51511 (19 pp.). https://doi.org/10.7554/eLife.51511
Verifying pore network models of imbibition in rocks using time-resolved synchrotron imaging
Bultreys, T., Singh, K., Raeini, A. Q., Ruspini, L. C., Øren, P. E., Berg, S., … Blunt, M. J. (2020). Verifying pore network models of imbibition in rocks using time-resolved synchrotron imaging. Water Resources Research, 56(6), e2019WR026587 (13 pp.). https://doi.org/10.1029/2019WR026587
Discovery of novel imidazopyridine GSK-3β inhibitors supported by cmputational approaches
Buonfiglio, R., Prati, F., Bischetti, M., Cavarischia, C., Furlotti, G., & Ombrato, R. (2020). Discovery of novel imidazopyridine GSK-3β inhibitors supported by cmputational approaches. Molecules, 25(9), 2163 (29 pp.). https://doi.org/10.3390/molecules25092163
Structural and functional insights into CWC27/CWC22 heterodimer linking the exon junction complex to spliceosomes
Busetto, V., Barbosa, I., Basquin, J., Marquenet, É., Hocq, R., Hennion, M., … Le Hir, H. (2020). Structural and functional insights into CWC27/CWC22 heterodimer linking the exon junction complex to spliceosomes. Nucleic Acids Research. https://doi.org/10.1093/nar/gkaa267
High-resolution crystal structures of a "half sandwich"-type Ru(II) coordination compound bound to hen egg-white lysozyme and proteinase K
Chiniadis, L., Bratsos, I., Bethanis, K., Karpusas, M., Giastas, P., & Papakyriakou, A. (2020). High-resolution crystal structures of a "half sandwich"-type Ru(II) coordination compound bound to hen egg-white lysozyme and proteinase K. Journal of Biological Inorganic Chemistry. https://doi.org/10.1007/s00775-020-01786-z
Structure of <em>Drosophila melanogaster</em> ARC1 reveals a repurposed molecule with characteristics of retroviral Gag
Cottee, M. A., Letham, S. C., Young, G. R., Stoye, J. P., & Taylor, I. A. (2020). Structure of Drosophila melanogaster ARC1 reveals a repurposed molecule with characteristics of retroviral Gag. Science Advances, 6(1), eaay6354 (12 pp.). https://doi.org/10.1126/sciadv.aay6354
How does successive hydrogen addition to PAH ions impact their unimolecular chemistry?
Diedhiou, M., West, B. J., & Mayer, P. M. (2020). How does successive hydrogen addition to PAH ions impact their unimolecular chemistry? Molecular Astrophysics, 19, 100071 (9 pp.). https://doi.org/10.1016/j.molap.2020.100071
Nucleosome-bound SOX2 and SOX11 structures elucidate pioneer factor function
Dodonova, S. O., Zhu, F., Dienemann, C., Taipale, J., & Cramer, P. (2020). Nucleosome-bound SOX2 and SOX11 structures elucidate pioneer factor function. Nature, 580(7805), 669-672. https://doi.org/10.1038/s41586-020-2195-y
Hybrid screening approach for very small fragments: X-ray and computational screening on FKBP51
Draxler, S. W., Bauer, M., Eickmeier, C., Nadal, S., Nar, H., Rangel Rojas, D., … Fiegen, D. (2020). Hybrid screening approach for very small fragments: X-ray and computational screening on FKBP51. Journal of Medicinal Chemistry, 63(11), 5856-5864. https://doi.org/10.1021/acs.jmedchem.0c00120
Structural basis for selectivity in a highly reducing type II polyketide synthase
Du, D., Katsuyama, Y., Horiuchi, M., Fushinobu, S., Chen, A., Davis, T. D., … Ohnishi, Y. (2020). Structural basis for selectivity in a highly reducing type II polyketide synthase. Nature Chemical Biology. https://doi.org/10.1038/s41589-020-0530-0
 

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