| Targeting cavity-creating p53 cancer mutations with small-molecule stabilizers: the Y220X paradigm
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| Electron and proton transfers modulate DNA binding by the transcription regulator RsrR
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| Structure-guided design of a peptide lock for modular peptide binders
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| In meso in situ serial X-Ray crystallography (IMISX): a protocol for membrane protein structure determination at the Swiss Light Source
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| Crystal structure of the translation recovery factor Trf from <em>Sulfolobus solfataricus</em>
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| A precisely positioned MED12 activation helix stimulates CDK8 kinase activity
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| Stereoselective activity of 1-propargyl-4-styrylpiperidine-like analogues that can discriminate between monoamine oxidase isoforms A and B
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| JUNGFRAU detector for brighter x-ray sources: solutions for IT and data science challenges in macromolecular crystallography
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| Human PLD structures enable drug design and characterization of isoenzyme selectivity
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| Ancestral-sequence reconstruction unveils the structural basis of function in mammalian FMOs
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| Structures of lipoprotein signal peptidase II from <em>Staphylococcus aureus</em> complexed with antibiotics globomycin and myxovirescin
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| Comparison of orexin 1 and orexin 2 ligand binding modes using X-ray crystallography and computational analysis
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| What does fluorine do to a protein? Thermodynamic, and highly-resolved structural insights into fluorine-labelled variants of the cold shock protein
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| Conformational changes in apolipoprotein N-acyltransferase (Lnt)
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| Discovery and optimization of heteroaryl piperazines as potent and selective PI3Kδ inhibitors
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| Fragment-based discovery of novel potent sepiapterin reductase inhibitors
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| Structure and function of photosystem I in <i>Cyanidioschyzon merolae</i>
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| Crystal structure of CC chemokine receptor 2A in complex with an orthosteric antagonist provides insights for the design of selective antagonists
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| Identification of 2-imidazopyridine and 2-aminopyridone purinones as potent pan-Janus kinase (JAK) inhibitors for the inhaled treatment of respiratory diseases
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| Structures in tetrahydrofolate methylation in desulfitobacterial glycine betaine metabolism at atomic resolution
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