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N‐terminal β‐strand in YAP is critical for stronger binding to scalloped relative to TEAD transcription factor
Fedir, B., Yannick, M., Marco, M., Patrizia, F., Catherine, Z., Frédéric, V., … Patrick, C. (2023). N‐terminal β‐strand in YAP is critical for stronger binding to scalloped relative to TEAD transcription factor. Protein Science, 32(1), e4545 (13 pp.). https://doi.org/10.1002/pro.4545
Optimization of a class of dihydrobenzofurane analogs toward orally efficacious YAP-TEAD protein-protein interaction inhibitors
Sellner, H., Chapeau, E., Furet, P., Voegtle, M., Salem, B., Le Douget, M., … Soldermann, N. (2023). Optimization of a class of dihydrobenzofurane analogs toward orally efficacious YAP-TEAD protein-protein interaction inhibitors. ChemMedChem, 18(11), e202300051 (23 pp.). https://doi.org/10.1002/cmdc.202300051
The first class of small molecules potently disrupting the YAP-TEAD interaction by direct competition
Furet, P., Bordas, V., Le Douget, M., Salem, B., Mesrouze, Y., Imbach-Weese, P., … Schmelzle, T. (2022). The first class of small molecules potently disrupting the YAP-TEAD interaction by direct competition. ChemMedChem, 17(19), e202200303 (14 pp.). https://doi.org/10.1002/cmdc.202200303
Identification of FAM181A and FAM181B as new interactors with the TEAD transcription factors
Bokhovchuk, F., Mesrouze, Y., Delaunay, C., Martin, T., Villard, F., Meyerhofer, M., … Chène, P. (2020). Identification of FAM181A and FAM181B as new interactors with the TEAD transcription factors. Protein Science, 29(2), 509-520. https://doi.org/10.1002/pro.3775
Molecular and structural characterization of a TEAD mutation at the origin of Sveinsson's chorioretinal atrophy
Bokhovchuk, F., Mesrouze, Y., Izaac, A., Meyerhofer, M., Zimmermann, C., Fontana, P., … Chène, P. (2019). Molecular and structural characterization of a TEAD mutation at the origin of Sveinsson's chorioretinal atrophy. FEBS Journal, 286(12), 2381-2398. https://doi.org/10.1111/febs.14817
Effect of the acylation of TEAD4 on its interaction with co-activators YAP and TAZ
Mesrouze, Y., Meyerhofer, M., Bokhovchuk, F., Fontana, P., Zimmermann, C., Martin, T., … Chène, P. (2017). Effect of the acylation of TEAD4 on its interaction with co-activators YAP and TAZ. Protein Science, 26(12), 2399-2409. https://doi.org/10.1002/pro.3312